µ-Conotoxins Targeting the Human Voltage-Gated Sodium Channel Subtype NaV1.7
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δ-conotoxin SuVIA suggests an evolutionary link between ancestral predator defence and the origin of fish-hunting behaviour in carnivorous cone snails
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Voltage-Gated Sodium Channel Modulation by a New Spider Toxin Ssp1a Isolated From an Australian Theraphosid
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Venom Peptides with Dual Modulatory Activity on the Voltage-Gated Sodium Channel NaV1.1 Provide Novel Leads for Development of Antiepileptic Drugs
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Venom chemistry underlying the painful stings of velvet ants (Hymenoptera: Mutillidae)
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Two for the Price of One: Heterobivalent Ligand Design Targeting Two Binding Sites on Voltage-Gated Sodium Channels Slows Ligand Dissociation and Enhances Potency
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Transfection methods for high-throughput cellular assays of voltage-gated calcium and sodium channels involved in pain
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The Snake with the Scorpion’s Sting: Novel Three-Finger Toxin Sodium Channel Activators from the Venom of the Long-Glanded Blue Coral Snake
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The E15R Point Mutation in Scorpion Toxin Cn2 Uncouples Its Depressant and Excitatory Activities on Human NaV1.6
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Synthesis of Pseudellone Analogs and Characterization as Novel T-type Calcium Channel Blockers
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Structural and functional insights into the inhibition of human voltage-gated sodium channels by μ-conotoxin KIIIA disulfide isomers
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Recombinant production, bioconjugation and membrane binding studies of Pn3a, a selective Nav1.7 inhibitor
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Recombinant Production , Bioconjugation and Membrane Binding Studies of Pn3a , a Selective Nav1.7 Inhibitor
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Rational engineering defines a molecular switch that is essential for activity of spider-venom peptides against the analgesics target Nav1.7
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Pharmacological screening technologies for venom peptide discovery
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Pharmacological Inhibition of the Voltage-Gated Sodium Channel NaV1.7 Alleviates Chronic Visceral Pain in a Rodent Model of Irritable Bowel Syndrome
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Pharmacological characterisation of the highly Nav1.7 selective spider venom peptide Pn3a
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Pharmacological activity and NMR solution structure of the leech peptide HSTX-I
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Pharmacological activity and NMR solution structure of the leech peptide HSTX-I
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Novel Neurotoxic Activity in Calliophis intestinalis Venom. Neurotoxicity Research
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Neurotoxic peptides from the venom of the giant Australian stinging tree
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Multiple sodium channel isoforms mediate the pathological effects of Pacific ciguatoxin-1
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Mapping the Molecular Surface of the Analgesic Nav1.7-Selective Peptide Pn3a Reveals Residues Essential for Membrane and Channel Interactions
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Manipulation of a spider peptide toxin alters its affinity for lipid bilayers and potency and selectivity for voltage-gated sodium channel subtype
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Identification and Characterization of ProTx-III [μ-TRTX-Tp1a], a New Voltage-Gated Sodium Channel Inhibitor from Venom of the Tarantula Thrixopelma pruriens
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Evaluation of Efficient Non-reducing Enzymatic and Chemical Ligation Strategies for Complex Disulfide-Rich Peptides
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Enzymatic Ligation of a Pore Blocker Toxin and a Gating Modifier Toxin: Creating Double-Knotted Peptides with Improved Sodium Channel Nav1.7 Inhibition
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Enzymatic Ligation of a Pore Blocker Toxin and a Gating Modifier Toxin: Creating Double-Knotted Peptides with Improved Sodium Channel Nav1.7 Inhibition
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Efficient Enzymatic Ligation of Inhibitor Cystine Knot Spider Venom Peptides: Using Sortase A To Form Double-Knottins That Probe Voltage-Gated Sodium Channel NaV1.7
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Discovery of Anti-tubercular Analogues of Bedaquiline with Modified A-, B-and C-Ring Subunits
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Discovery and mode of action of a novel analgesic β-toxin from the African spider Ceratogyrus darlingi
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Diindolylmethane Derivatives: New Selective Blockers for T-Type Calcium Channels
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Development of a high-throughput fluorescent no-wash sodium influx assay
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Characterization of Synthetic Tf2 as a Nav1.3 Selective Pharmacological Probe
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Characterization of Synthetic Tf2 as a Nav1.3 Selective Pharmacological Probe
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Characterisation of δ-Conotoxin TxVIA as a Mammalian T-Type Calcium Channel Modulator
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Analgesic Effects of GpTx-1, PF-04856264 and CNV1014802 in a Mouse Model of Nav1.7-Mediated Pain
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A spider-venom peptide with multitarget activity on sodium and calcium channels alleviates chronic visceral pain in a model of irritable bowel syndrome
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A Selective Nav1.1 Activator with Potential for Treatment of Dravet Syndrome Epilepsy
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A Selective Nav1.1 Activator with Potential for Treatment of Dravet Syndrome Epilepsy
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A comprehensive portrait of the venom of the giant red bull ant, Myrmecia gulosa, reveals a hyperdiverse hymenopteran toxin gene family
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